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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50162753(1-(4-But-2-ynyloxy-benzenesulfonyl)-[1,4]diazepane...)
Affinity DataIC50:  11nMAssay Description:Inhibitory concentration against TNF-alpha converting enzyme at 1 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50162753(1-(4-But-2-ynyloxy-benzenesulfonyl)-[1,4]diazepane...)
Affinity DataIC50:  225nMAssay Description:Inhibitory concentration against Matrix metalloproteinase-13 at 1 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50162753(1-(4-But-2-ynyloxy-benzenesulfonyl)-[1,4]diazepane...)
Affinity DataIC50:  576nMAssay Description:Inhibitory concentration against matrix metalloproteinase-1 at 1 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed