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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 6 hits in this display   

TargetBromodomain-containing protein 2(Homo sapiens (Human))TBA
LigandPNGBDBM50481804(CHEMBL5281933)
Affinity DataKd:  111nMAssay Description:Binding affinity to BRD2 BD1 domain (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))TBA
LigandPNGBDBM50481804(CHEMBL5281933)
Affinity DataKd:  94nMAssay Description:Binding affinity to BRD2 BD2 domain (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM50481804(CHEMBL5281933)
Affinity DataKd:  44nMAssay Description:Binding affinity to BRD4 BD2 domain (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))TBA
LigandPNGBDBM50481804(CHEMBL5281933)
Affinity DataKd:  39nMAssay Description:Binding affinity to BRD3 BD2 domain (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM50481804(CHEMBL5281933)
Affinity DataKd:  75nMAssay Description:Binding affinity to BRD4 BD1 domain (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))TBA
LigandPNGBDBM50481804(CHEMBL5281933)
Affinity DataKd:  35nMAssay Description:Binding affinity to BRD3 BD1 domain (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed