Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetCathepsin K(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50129071(Acetic acid (1S,2S,4R)-3-[(2-benzyloxycarbonylamin...)
Affinity DataKi:  8.80nMAssay Description:Inhibitory activity of the compound was measured against Cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50129071(Acetic acid (1S,2S,4R)-3-[(2-benzyloxycarbonylamin...)
Affinity DataKi:  130nMAssay Description:Inhibitory activity of the compound was measured against Cathepsin SMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50129071(Acetic acid (1S,2S,4R)-3-[(2-benzyloxycarbonylamin...)
Affinity DataKi:  1.60E+3nMAssay Description:Inhibitory activity of the compound was measured against Cathepsin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50129071(Acetic acid (1S,2S,4R)-3-[(2-benzyloxycarbonylamin...)
Affinity DataKi:  3.70E+3nMAssay Description:Inhibitory activity of the compound was measured against Cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed