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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 12 hits in this display   

TargetNeutrophil collagenase(Homo sapiens (Human))
University Hospital M£Nster

Curated by ChEMBL
LigandPNGBDBM50225397((R)-2-(N-benzyl-4-(2-fluoroethoxy)phenylsulfonamid...)
Affinity DataIC50:  2nMAssay Description:Inhibition of MMP8 using (7-methoxycoumarin-4-yl)acetyl-Pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl)-L-2,3-diaminopropionyl)Ala-Arg-NH2 as substrate incuba...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil collagenase(Homo sapiens (Human))
University Hospital M£Nster

Curated by ChEMBL
LigandPNGBDBM50225397((R)-2-(N-benzyl-4-(2-fluoroethoxy)phenylsulfonamid...)
Affinity DataIC50:  2nMAssay Description:Inhibition of MMP8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil collagenase(Homo sapiens (Human))
University Hospital M£Nster

Curated by ChEMBL
LigandPNGBDBM50225397((R)-2-(N-benzyl-4-(2-fluoroethoxy)phenylsulfonamid...)
Affinity DataIC50:  2nMAssay Description:Inhibition of MMP-8 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
University Hospital Of The Westf£Lische Wilhelms-Universit£T M£Nster

Curated by ChEMBL
LigandPNGBDBM50225397((R)-2-(N-benzyl-4-(2-fluoroethoxy)phenylsulfonamid...)
Affinity DataIC50:  4nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
University Hospital Of The Westf£Lische Wilhelms-Universit£T M£Nster

Curated by ChEMBL
LigandPNGBDBM50225397((R)-2-(N-benzyl-4-(2-fluoroethoxy)phenylsulfonamid...)
Affinity DataIC50:  4nMAssay Description:Inhibition of MMP-2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
University Hospital Of The Westf£Lische Wilhelms-Universit£T M£Nster

Curated by ChEMBL
LigandPNGBDBM50225397((R)-2-(N-benzyl-4-(2-fluoroethoxy)phenylsulfonamid...)
Affinity DataIC50:  4nMAssay Description:Inhibition of MMP2 using (7-methoxycoumarin-4-yl)acetyl-Pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl)-L-2,3-diaminopropionyl)Ala-Arg-NH2 as substrate incuba...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
University Hospital Of The Westf£Lische Wilhelms-Universit£T M£Nster

Curated by ChEMBL
LigandPNGBDBM50225397((R)-2-(N-benzyl-4-(2-fluoroethoxy)phenylsulfonamid...)
Affinity DataIC50:  11nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
University Hospital Of The Westf£Lische Wilhelms-Universit£T M£Nster

Curated by ChEMBL
LigandPNGBDBM50225397((R)-2-(N-benzyl-4-(2-fluoroethoxy)phenylsulfonamid...)
Affinity DataIC50:  11nMAssay Description:Inhibition of MMP13 using (7-methoxycoumarin-4-yl)acetyl-Pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl)-L-2,3-diaminopropionyl)Ala-Arg-NH2 as substrate incub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
University Hospital Of The Westf£Lische Wilhelms-Universit£T M£Nster

Curated by ChEMBL
LigandPNGBDBM50225397((R)-2-(N-benzyl-4-(2-fluoroethoxy)phenylsulfonamid...)
Affinity DataIC50:  11nMAssay Description:Inhibition of MMP-13 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
University Hospital M£Nster

Curated by ChEMBL
LigandPNGBDBM50225397((R)-2-(N-benzyl-4-(2-fluoroethoxy)phenylsulfonamid...)
Affinity DataIC50:  50nMAssay Description:Inhibition of MMP-9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
University Hospital M£Nster

Curated by ChEMBL
LigandPNGBDBM50225397((R)-2-(N-benzyl-4-(2-fluoroethoxy)phenylsulfonamid...)
Affinity DataIC50:  50nMAssay Description:Inhibition of MMP9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
University Hospital M£Nster

Curated by ChEMBL
LigandPNGBDBM50225397((R)-2-(N-benzyl-4-(2-fluoroethoxy)phenylsulfonamid...)
Affinity DataIC50:  50nMAssay Description:Inhibition of MMP9 using (7-methoxycoumarin-4-yl)acetyl-Pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl)-L-2,3-diaminopropionyl)Ala-Arg-NH2 as substrate incuba...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed