Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 10 hits in this display
Caspase-3(Homo sapiens (Human))Novagenesis Foundation
US Patent
BDBM160796(US10167313, Compound 63 | US9045524, 63)
Caspase-3(Homo sapiens (Human))Novagenesis Foundation
US Patent
BDBM160796(US10167313, Compound 63 | US9045524, 63)
Caspase-7(Homo sapiens (Human))Novagenesis Foundation
US Patent
BDBM160796(US10167313, Compound 63 | US9045524, 63)
Caspase-7(Homo sapiens (Human))Novagenesis Foundation
US Patent
BDBM160796(US10167313, Compound 63 | US9045524, 63)
IC50: 1.80E+3nMAssay Description:Selectivity of compound 55, compound 63, compound 48, compound 57, compound 88 toward caspase-1 (pro-inflammatory group), caspase-5 (group I), caspas...More data for this Ligand-Target Pair
Caspase-9(Homo sapiens (Human))Novagenesis Foundation
US Patent
BDBM160796(US10167313, Compound 63 | US9045524, 63)
IC50: >3.33E+3nMT: 2°CAssay Description:Selectivity of compound 55, compound 63, compound 48, compound 57, compound 88 toward caspase-1 (pro-inflammatory group), caspase-5 (group I), caspas...More data for this Ligand-Target Pair
Caspase-9(Homo sapiens (Human))Novagenesis Foundation
US Patent
BDBM160796(US10167313, Compound 63 | US9045524, 63)
IC50: >3.33E+3nMAssay Description:Selectivity of compound 55, compound 63, compound 48, compound 57, compound 88 toward caspase-1 (pro-inflammatory group), caspase-5 (group I), caspas...More data for this Ligand-Target Pair
Caspase-1(Homo sapiens (Human))Genesis Technologies
US Patent
BDBM160796(US10167313, Compound 63 | US9045524, 63)
IC50: >3.33E+3nMAssay Description:Selectivity of compound 55, compound 63, compound 48, compound 57, compound 88 toward caspase-1 (pro-inflammatory group), caspase-5 (group I), caspas...More data for this Ligand-Target Pair
Caspase-5(Homo sapiens (Human))Genesis Technologies
US Patent
BDBM160796(US10167313, Compound 63 | US9045524, 63)
IC50: >3.33E+3nMAssay Description:Selectivity of compound 55, compound 63, compound 48, compound 57, compound 88 toward caspase-1 (pro-inflammatory group), caspase-5 (group I), caspas...More data for this Ligand-Target Pair
Caspase-5(Homo sapiens (Human))Genesis Technologies
US Patent
BDBM160796(US10167313, Compound 63 | US9045524, 63)
IC50: >3.33E+3nMT: 2°CAssay Description:Selectivity of compound 55, compound 63, compound 48, compound 57, compound 88 toward caspase-1 (pro-inflammatory group), caspase-5 (group I), caspas...More data for this Ligand-Target Pair
Caspase-1(Homo sapiens (Human))Genesis Technologies
US Patent
BDBM160796(US10167313, Compound 63 | US9045524, 63)
IC50: >3.33E+3nMT: 2°CAssay Description:Selectivity of compound 55, compound 63, compound 48, compound 57, compound 88 toward caspase-1 (pro-inflammatory group), caspase-5 (group I), caspas...More data for this Ligand-Target Pair