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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
hits in this display
Target
Motilin receptor
(Homo sapiens (Human))
Tranzyme Pharma
Curated by
ChEMBL
Ligand
BDBM50214272
((5R,8R,11S)-11-(aminomethyl)-8-(propan-2-yl)-5-{[3...)
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Affinity Data
Ki: 15nM
Assay Description:
Displacement of [125I]-motilin from human motilin receptor expressed in CHO cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
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Target
Motilin receptor
(Homo sapiens (Human))
Tranzyme Pharma
Curated by
ChEMBL
Ligand
BDBM50214272
((5R,8R,11S)-11-(aminomethyl)-8-(propan-2-yl)-5-{[3...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 8nM
Assay Description:
Antagonist activity against human motilin receptor in aequoscreen cells assessed as inhibition of motilin induced calcium release by aequorin assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI