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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Westf£Lische Wilhelms-Universit£T

Curated by ChEMBL
LigandPNGBDBM50500713(CHEMBL3752747)
Affinity DataIC50:  393nMAssay Description:Inhibition of human MMP9 using (7-methoxycoumarin-4-yl) acetyl pro-Leu-Gly-Leu-[3-(2,4-dinitrophenyl)-L-2,3-diamino-propionyl]-Ala-Arg-NH2 as substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Westf£Lische Wilhelms-Universit£T

Curated by ChEMBL
LigandPNGBDBM50500713(CHEMBL3752747)
Affinity DataIC50:  628nMAssay Description:Inhibition of human MMP2 using (7-methoxycoumarin-4-yl) acetyl pro-Leu-Gly-Leu-[3-(2,4-dinitrophenyl)-L-2,3-diamino-propionyl]-Ala-Arg-NH2 as substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Westf£Lische Wilhelms-Universit£T

Curated by ChEMBL
LigandPNGBDBM50500713(CHEMBL3752747)
Affinity DataIC50:  1.03E+3nMAssay Description:Inhibition of MMP13 (unknown origin) using (7-methoxycoumarin-4-yl) acetyl pro-Leu-Gly-Leu-[3-(2,4-dinitrophenyl)-L-2,3-diamino-propionyl]-Ala-Arg-NH...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeutrophil collagenase(Homo sapiens (Human))
Westf£Lische Wilhelms-Universit£T

Curated by ChEMBL
LigandPNGBDBM50500713(CHEMBL3752747)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of MMP8 (unknown origin) using (7-methoxycoumarin-4-yl) acetyl pro-Leu-Gly-Leu-[3-(2,4-dinitrophenyl)-L-2,3-diamino-propionyl]-Ala-Arg-NH2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed