Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetEndothelin-converting enzyme 1(Bos taurus)
TBA

Curated by ChEMBL

LigandBDBM50282595(CHEMBL281562 | PO3 2-Leu-Trp-O-3K)Copy SMILESCopy InChI

Affinity DataIC50:  960nMAssay Description:Inhibition of Endothelin-converting enzyme (ECE) from microsomal fractions of bovine cultured endothelial cellsMore data for this Ligand-Target Pair

Target InfoPDBMMDB
UniProtKB/SwissProt
B.MOADGoogleScholar

Ligand InfoCHEMBLKEGGPC cidPC sidSimilars

In DepthDetails Article
Copy BDB DOI

TargetEndothelin-converting enzyme 1(Homo sapiens (Human))
TBA

Curated by ChEMBL

LigandBDBM50287436((S)-3-(1H-Indol-3-yl)-2-((S)-4-methyl-2-phosphonoa...)Copy SMILESCopy InChI

Affinity DataIC50:  1.50E+3nMAssay Description:In vitro inhibition of phosphoramidon-sensitive membrane bound zinc metalloprotease Endothelin-converting enzyme from partially purified guinea pig l...More data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoCHEMBLKEGGPC cidPC sidSimilars

In DepthDetails Article
Copy BDB DOI