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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 8 hits in this display   

TargetMatrix metalloproteinase-9(Mus musculus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50078568((S)-4-Benzylsulfanyl-2-[(biphenyl-4-sulfonyl)-isob...)
Affinity DataIC50:  2.5nMAssay Description:Inhibitory concentration required against matrix metalloprotease-9 (MMP-9 gelatinase B)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50103995(4-Benzylsulfanyl-2-[(biphenyl-4-sulfonyl)-isobutyl...)
Affinity DataIC50:  2.5nMAssay Description:In vitro inhibition of human matrix metalloprotease-9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50103995(4-Benzylsulfanyl-2-[(biphenyl-4-sulfonyl)-isobutyl...)
Affinity DataIC50:  3.80nMAssay Description:In vitro inhibition of human matrix metalloprotease-13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50078568((S)-4-Benzylsulfanyl-2-[(biphenyl-4-sulfonyl)-isob...)
Affinity DataIC50:  3.80nMAssay Description:Inhibition of matrix metalloprotease-13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50103995(4-Benzylsulfanyl-2-[(biphenyl-4-sulfonyl)-isobutyl...)
Affinity DataIC50:  4.10nMAssay Description:In vitro inhibition of human matrix metalloprotease-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Mus musculus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50078568((S)-4-Benzylsulfanyl-2-[(biphenyl-4-sulfonyl)-isob...)
Affinity DataIC50:  4.10nMAssay Description:Inhibition of matrix metalloprotease-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50078568((S)-4-Benzylsulfanyl-2-[(biphenyl-4-sulfonyl)-isob...)
Affinity DataIC50:  90nMAssay Description:Inhibition of matrix metalloprotease-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50103995(4-Benzylsulfanyl-2-[(biphenyl-4-sulfonyl)-isobutyl...)
Affinity DataIC50:  90nMAssay Description:In vitro inhibitory activity against matrix metalloprotease-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed