Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50139823(10-Chloro-6-hydroxy-5-isobutyl-pyrido[1,2-a]quinol...)
Affinity DataEC50:  2.60E+4nMAssay Description:Half-Maximal effective concentration of compound required to stimulate of wild type-CFTR activity in the presence of 10 microM FskMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50139823(10-Chloro-6-hydroxy-5-isobutyl-pyrido[1,2-a]quinol...)
Affinity DataEC50:  3.20E+4nMAssay Description:Half-Maximal effective concentration of compound required to stimulate of G551D-CFTR activity in the presence of 10 microM FskMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed