Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL

LigandBDBM50033418(CHEMBL3357685)Copy SMILESCopy InChI

Affinity DataIC50:  4nMAssay Description:Inhibition of human N-myristoyltransferase 1 assessed as transfer of [3H]-myristic acid to a biotinylated substrate peptide (GCGGSKVKPQPPQAK(biotin)-...More data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoPurchaseCHEMBLPC cidPC sidPDBSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetGlycylpeptide N-tetradecanoyltransferase(Aspergillus fumigatus)
Temple University

Curated by ChEMBL

LigandBDBM50033418(CHEMBL3357685)Copy SMILESCopy InChI

Affinity DataIC50:  12nMAssay Description:Inhibition of recombinant Aspergillus fumigatus NMT (Gln86 to Leu492 residues) expressed in Escherichia coli BL21(DE3) pLysS cells using [3H]-myristo...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPurchaseCHEMBLPC cidPC sidPDBSimilars

In DepthDetails ArticlePubMedPDB3D Structure (crystal)
Copy BDB DOI