Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 11 hits in this display   

TargetHistone deacetylase 6(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50008222(CHEMBL3235118)
Affinity DataIC50:  12nMAssay Description:Inhibition of human HDAC-6 using RHKK(Ac) as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50008222(CHEMBL3235118)
Affinity DataIC50:  31nMAssay Description:Displacement of GM-FITC from full-length recombinant human Hsp90-alpha after 4 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50008222(CHEMBL3235118)
Affinity DataIC50:  717nMAssay Description:Inhibition of human HDAC-8 using RHKK(Ac) as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 11(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50008222(CHEMBL3235118)
Affinity DataIC50:  1.77E+3nMAssay Description:Inhibition of human HDAC-11 using RHKK(Ac) as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 5(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50008222(CHEMBL3235118)
Affinity DataIC50:  1.91E+3nMAssay Description:Inhibition of human HDAC-5 using RHKK(Ac) as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3/Nuclear receptor corepressor 2 (HDAC3/NCoR2)(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50008222(CHEMBL3235118)
Affinity DataIC50:  2.79E+3nMAssay Description:Inhibition of human HDAC-3/NCOR2 using RHKK(Ac) as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50008222(CHEMBL3235118)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition of human HDAC-1 using RHKK(Ac) as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyamine deacetylase HDAC10(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50008222(CHEMBL3235118)
Affinity DataIC50:  3.22E+3nMAssay Description:Inhibition of human HDAC-10 using RHKK(Ac) as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50008222(CHEMBL3235118)
Affinity DataIC50:  5.61E+3nMAssay Description:Inhibition of human HDAC-2 using RHKK(Ac) as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 7(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50008222(CHEMBL3235118)
Affinity DataIC50:  4.55E+4nMAssay Description:Inhibition of human HDAC-7 using RHKK(Ac) as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50008222(CHEMBL3235118)
Affinity DataIC50:  7.15E+4nMAssay Description:Inhibition of human HDAC-4 using RHKK(Ac) as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed