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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
12
hits in this display
Target
Lysine-specific demethylase 5B
(Homo sapiens (Human))
Celgene Quanticel Research
US Patent
Ligand
BDBM270504
(3-{[((1S)-5-{methyl[4-(methylethyl)phenyl]amino}is...)
Copy SMILES
Copy InChI
Affinity Data
IC50: <100nM
Assay Description:
Jarid1b: The ability of test compounds to inhibit the activity of Jarid1B was determined in 384-well plate format under the following reaction condit...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Lysine-specific demethylase 5B
(Homo sapiens (Human))
Celgene Quanticel Research
US Patent
Ligand
BDBM270504
(3-{[((1S)-5-{methyl[4-(methylethyl)phenyl]amino}is...)
Copy SMILES
Copy InChI
Affinity Data
IC50: <100nM
Assay Description:
Jarid1b: The ability of test compounds to inhibit the activity of Jarid1B was determined in 384-well plate format under the following reaction condit...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Lysine-specific demethylase 5B
(Homo sapiens (Human))
Celgene Quanticel Research
US Patent
Ligand
BDBM270504
(3-{[((1S)-5-{methyl[4-(methylethyl)phenyl]amino}is...)
Copy SMILES
Copy InChI
Affinity Data
IC50: <100nM
Assay Description:
The ability of test compounds to inhibit the activity of Jarid1B was determined in 384-well plate format under the following reaction conditions: 0.8...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Lysine-specific demethylase 5B
(Homo sapiens (Human))
Celgene Quanticel Research
US Patent
Ligand
BDBM270504
(3-{[((1S)-5-{methyl[4-(methylethyl)phenyl]amino}is...)
Copy SMILES
Copy InChI
Affinity Data
IC50: <100nM
Assay Description:
The ability of test compounds to inhibit the activity of Jarid1B was determined in 384-well plate format under the following reaction conditions: 0.8...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Lysine-specific demethylase 6B
(Homo sapiens (Human))
Celgene Quanticel Research
US Patent
Ligand
BDBM270504
(3-{[((1S)-5-{methyl[4-(methylethyl)phenyl]amino}is...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 5.50E+3nM
Assay Description:
JMJD3: The enzymatic assay of JMJD3 activity is based upon Time Resolved-Fluorescence Resonance Energy Transfer (TR-FRET) detection. The ability of t...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Lysine-specific demethylase 4C
(Homo sapiens (Human))
Celgene Quanticel Research
US Patent
Ligand
BDBM270504
(3-{[((1S)-5-{methyl[4-(methylethyl)phenyl]amino}is...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 5.50E+3nM
Assay Description:
The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Lysine-specific demethylase 4C
(Homo sapiens (Human))
Celgene Quanticel Research
US Patent
Ligand
BDBM270504
(3-{[((1S)-5-{methyl[4-(methylethyl)phenyl]amino}is...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 5.50E+3nM
Assay Description:
JMJD2C: The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditio...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Lysine-specific demethylase 6B
(Homo sapiens (Human))
Celgene Quanticel Research
US Patent
Ligand
BDBM270504
(3-{[((1S)-5-{methyl[4-(methylethyl)phenyl]amino}is...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 5.50E+3nM
Assay Description:
JMJD3: The enzymatic assay of JMJD3 activity is based upon Time Resolved-Fluorescence Resonance Energy Transfer (TR-FRET) detection. The ability of t...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Lysine-specific demethylase 4C
(Homo sapiens (Human))
Celgene Quanticel Research
US Patent
Ligand
BDBM270504
(3-{[((1S)-5-{methyl[4-(methylethyl)phenyl]amino}is...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 5.50E+3nM
Assay Description:
JMJD2C: The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditio...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Lysine-specific demethylase 6B
(Homo sapiens (Human))
Celgene Quanticel Research
US Patent
Ligand
BDBM270504
(3-{[((1S)-5-{methyl[4-(methylethyl)phenyl]amino}is...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 5.50E+3nM
Assay Description:
The enzymatic assay of JMJD3 activity is based upon Time Resolved-Fluorescence Resonance Energy Transfer (TR-FRET) detection. The ability of test com...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Lysine-specific demethylase 6B
(Homo sapiens (Human))
Celgene Quanticel Research
US Patent
Ligand
BDBM270504
(3-{[((1S)-5-{methyl[4-(methylethyl)phenyl]amino}is...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 5.50E+3nM
Assay Description:
The enzymatic assay of JMJD3 activity is based upon Time Resolved-Fluorescence Resonance Energy Transfer (TR-FRET) detection. The ability of test com...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Lysine-specific demethylase 4C
(Homo sapiens (Human))
Celgene Quanticel Research
US Patent
Ligand
BDBM270504
(3-{[((1S)-5-{methyl[4-(methylethyl)phenyl]amino}is...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 5.50E+3nM
Assay Description:
The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI