Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 7 hits in this display
BDBM26793(benzimidazole analog., 19 | tert-butyl (3S,4S)-3-(...)
Matrilysin(Homo sapiens (Human))Bristol-Myers Squibb
BDBM26793(benzimidazole analog., 19 | tert-butyl (3S,4S)-3-(...)
BDBM26793(benzimidazole analog., 19 | tert-butyl (3S,4S)-3-(...)
Ki: 3.92E+3nM ΔG°: -30.9kJ/molepH: 7.5 T: 2°CAssay Description:The compounds were tested for enzyme inhibition using fluorescence resonance energy transfer (FRET) assay. Fluorescence measurements were performed i...More data for this Ligand-Target Pair
BDBM26793(benzimidazole analog., 19 | tert-butyl (3S,4S)-3-(...)
Ki: >5.03E+3nMAssay Description:The compounds were tested for enzyme inhibition using fluorescence resonance energy transfer (FRET) assay. Fluorescence measurements were performed i...More data for this Ligand-Target Pair
BDBM26793(benzimidazole analog., 19 | tert-butyl (3S,4S)-3-(...)
IC50: 1nMpH: 7.5 T: 2°CAssay Description:The compounds were tested for enzyme inhibition using fluorescence resonance energy transfer (FRET) assay. Fluorescence measurements were performed i...More data for this Ligand-Target Pair
BDBM26793(benzimidazole analog., 19 | tert-butyl (3S,4S)-3-(...)
IC50: 390nMpH: 7.5 T: 2°CAssay Description:The compounds were tested for enzyme inhibition using fluorescence resonance energy transfer (FRET) assay. Fluorescence measurements were performed i...More data for this Ligand-Target Pair
BDBM26793(benzimidazole analog., 19 | tert-butyl (3S,4S)-3-(...)
IC50: 4.60E+3nMAssay Description:The compounds were tested for enzyme inhibition using fluorescence resonance energy transfer (FRET) assay. Fluorescence measurements were performed i...More data for this Ligand-Target Pair