Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetPoly [ADP-ribose] polymerase 2(Mus musculus (Mouse))
Nirma University

Curated by ChEMBL
LigandPNGBDBM50536937(CHEMBL4554200)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of mouse recombinant PARP2 by chemiluminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Nirma University

Curated by ChEMBL
LigandPNGBDBM50536937(CHEMBL4554200)
Affinity DataIC50:  5.40nMAssay Description:Inhibition of human recombinant PARP1 by chemiluminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Homo sapiens (Human))
Nirma University

Curated by ChEMBL
LigandPNGBDBM50536937(CHEMBL4554200)
Affinity DataIC50:  133nMAssay Description:Inhibition of human recombinant TNKS1 by chemiluminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
Nirma University

Curated by ChEMBL
LigandPNGBDBM50536937(CHEMBL4554200)
Affinity DataIC50:  290nMAssay Description:Inhibition of human recombinant TNKS2 by chemiluminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed