Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetLysophosphatidic acid receptor 1(Rattus norvegicus)
Ajinomoto

Curated by ChEMBL

LigandBDBM50211654(5-(4-(4-((1-(2-chlorophenyl)ethoxy)carbonyl)isoxaz...)Copy SMILESCopy InChI

Affinity DataIC50:  120nMAssay Description:Antagonist activity at LPA1 receptor in rat hepatic stellate cells assessed as inhibition of lysophosphatidic acid-induced intracellular calcium infl...More data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidPatentsSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
Ajinomoto

Curated by ChEMBL

LigandBDBM50211654(5-(4-(4-((1-(2-chlorophenyl)ethoxy)carbonyl)isoxaz...)Copy SMILESCopy InChI

Affinity DataIC50:  370nMAssay Description:Antagonist activity at human recombinant LPA1 receptor expressed in CHOK1 cells assessed as inhibition of lysophosphatidic acid-induced intracellular...More data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidPatentsSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI