Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetChymase(Homo sapiens (Human))
Daiichi Sankyo

US Patent
LigandPNGBDBM100746(US8507714, 150 | US8507714, 277)
Affinity DataIC50:  140nMAssay Description:Inhibitory activity of the compounds for recombinant human chymase was measured by method of Pasztor et al. (Pasztor et al., Acta Biol. Hung. 42:285-...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetChymase(Homo sapiens (Human))
Daiichi Sankyo

US Patent
LigandPNGBDBM100746(US8507714, 150 | US8507714, 277)
Affinity DataIC50:  160nMAssay Description:Inhibitory activity of the compounds for recombinant human chymase was measured by method of Pasztor et al. (Pasztor et al., Acta Biol. Hung. 42:285-...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetChymase(Homo sapiens (Human))
Daiichi Sankyo

US Patent
LigandPNGBDBM100748(CHEMBL246560 | US8507714, 277)
Affinity DataIC50:  170nMAssay Description:Inhibition of human recombinant chymaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin G(Homo sapiens (Human))
Daiichi Asubio Pharma

Curated by ChEMBL
LigandPNGBDBM100748(CHEMBL246560 | US8507714, 277)
Affinity DataIC50:  2.80E+4nMAssay Description:Inhibition of human cathepsin GMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed