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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 8 hits in this display   

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Homo sapiens (Human))
University Health Network

Curated by ChEMBL
LigandPNGBDBM50426302(CHEMBL2312698)
Affinity DataKi:  1.31E+5nMAssay Description:Inhibition of PAD4 (unknown origin) at 37 degCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-arginine deiminase type-2(Mus musculus)
University Health Network

Curated by ChEMBL
LigandPNGBDBM50426302(CHEMBL2312698)
Affinity DataKi:  1.79E+5nMAssay Description:Inhibition of full length recombinant mouse N-terminal GST-tagged PAD2 expressed in baculovirus infected Sf9 cells using benzoyl arginine ethyl ester...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-arginine deiminase type-4(Homo sapiens (Human))
University Health Network

Curated by ChEMBL
LigandPNGBDBM50426302(CHEMBL2312698)
Affinity DataKi:  1.83E+5nMAssay Description:Inhibition of full length recombinant human N-terminal GST-tagged PAD4 expressed in baculovirus infected Sf9 cells using benzoyl arginine ethylester ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Homo sapiens (Human))
University Health Network

Curated by ChEMBL
LigandPNGBDBM50426302(CHEMBL2312698)
Affinity DataKi:  3.71E+5nMAssay Description:Inhibition of PAD4 (unknown origin) at 52 degCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-arginine deiminase type-1(Homo sapiens (Human))
University Health Network

Curated by ChEMBL
LigandPNGBDBM50426302(CHEMBL2312698)
Affinity DataKi:  4.45E+5nMAssay Description:Inhibition of human PAD1 using BAEE as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Zhejiang Ocean University

Curated by ChEMBL
LigandPNGBDBM50426302(CHEMBL2312698)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of PDE4 (unknown origin) by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Homo sapiens (Human))
University Health Network

Curated by ChEMBL
LigandPNGBDBM50426302(CHEMBL2312698)
Affinity DataIC50:  1.38E+6nMAssay Description:Inhibition of PAD4 (unknown origin) at 37 degCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Homo sapiens (Human))
University Health Network

Curated by ChEMBL
LigandPNGBDBM50426302(CHEMBL2312698)
Affinity DataIC50:  4.27E+6nMAssay Description:Inhibition of PAD4 (unknown origin) at 52 degCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed