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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 6 hits in this display   

Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis)
The University Of Birmingham

Curated by ChEMBL
LigandPNGBDBM50134358(3,5-dimethyl-4-hydroxy-5-(4-methylbenzyl)-5H-thiop...)
Affinity DataIC50:  1.12E+5nMAssay Description:In vitro inhibitory activity against the recombinant Mycobacterium tuberculosis Beta-ketoacyl-ACP synthase III mtFabH condensing enzyme.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Escherichia coli)
National Institute Of Allergy And Infectious Diseases

Curated by ChEMBL
LigandPNGBDBM50134358(3,5-dimethyl-4-hydroxy-5-(4-methylbenzyl)-5H-thiop...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory activity against FabH from Escherichia coli ANSIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 1(Escherichia coli (strain K12))
National Institute Of Allergy And Infectious Diseases

Curated by ChEMBL
LigandPNGBDBM50134358(3,5-dimethyl-4-hydroxy-5-(4-methylbenzyl)-5H-thiop...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory activity against FabB from Escherichia coli ANSIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 2(Mycobacterium tuberculosis)
National Institute Of Allergy And Infectious Diseases

Curated by ChEMBL
LigandPNGBDBM50134358(3,5-dimethyl-4-hydroxy-5-(4-methylbenzyl)-5H-thiop...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory activity against KasB from Mycobacterium tuberculosis H37RvMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis)
The University Of Birmingham

Curated by ChEMBL
LigandPNGBDBM50134358(3,5-dimethyl-4-hydroxy-5-(4-methylbenzyl)-5H-thiop...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory activity against FabH from Mycobacterium tuberculosis H37RvMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis)
The University Of Birmingham

Curated by ChEMBL
LigandPNGBDBM50134358(3,5-dimethyl-4-hydroxy-5-(4-methylbenzyl)-5H-thiop...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory activity against KasA from Mycobacterium tuberculosis H37RvMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed