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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetAdenosine kinase(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50095367(5-(2,3-Dimethyl-cyclohexyl)-7-(6-morpholin-4-yl-py...)
Affinity DataIC50:  0.230nMAssay Description:Inhibitory activity against cytosolic adenosine kinase by ADO phosphorylation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50095367(5-(2,3-Dimethyl-cyclohexyl)-7-(6-morpholin-4-yl-py...)
Affinity DataIC50:  102nMAssay Description:Inhibitory activity against intact cell adenosine kinase by ADO phosphorylation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed