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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
8
hits in this display
Target
Mu-type opioid receptor
(Rattus norvegicus (rat))
R. W. Johnson Pharmaceutical Research Institute
Curated by
PDSP K
i
Database
Ligand
BDBM82269
((+)-alpha-Propoxyphene | CAS_469-62-5 | PROPOXYPHE...)
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Affinity Data
Ki: 34.5nM
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
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Target
Delta-type opioid receptor
(Rattus norvegicus (rat))
R. W. Johnson Pharmaceutical Research Institute
Curated by
PDSP K
i
Database
Ligand
BDBM82269
((+)-alpha-Propoxyphene | CAS_469-62-5 | PROPOXYPHE...)
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Affinity Data
Ki: 380nM
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
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Target
Kappa-type opioid receptor
(Rattus norvegicus (rat))
R. W. Johnson Pharmaceutical Research Institute
Curated by
PDSP K
i
Database
Ligand
BDBM82269
((+)-alpha-Propoxyphene | CAS_469-62-5 | PROPOXYPHE...)
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Affinity Data
Ki: 1.22E+3nM
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
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Target
Sodium-dependent serotonin transporter
(Rattus norvegicus (rat))
R. W. Johnson Pharmaceutical Research Institute
Curated by
PDSP K
i
Database
Ligand
BDBM82269
((+)-alpha-Propoxyphene | CAS_469-62-5 | PROPOXYPHE...)
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Affinity Data
Ki: >1.00E+4nM
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
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Target
Norepinephrine transporter
(RAT)
R. W. Johnson Pharmaceutical Research Institute
Curated by
PDSP K
i
Database
Ligand
BDBM82269
((+)-alpha-Propoxyphene | CAS_469-62-5 | PROPOXYPHE...)
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Affinity Data
Ki: >1.00E+4nM
More data for this Ligand-Target Pair
Target Info
UniProtKB/TrEMBL
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Target
Potassium voltage-gated channel subfamily H member 2
(Homo sapiens (Human))
Tcg Lifesciences
Curated by
ChEMBL
Ligand
BDBM82269
((+)-alpha-Propoxyphene | CAS_469-62-5 | PROPOXYPHE...)
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Affinity Data
IC50: 2.75E+3nM
Assay Description:
Inhibition of human ERG
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
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ChEBI
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Article
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Target
Mas-related G-protein coupled receptor member X2
(Homo sapiens (Human))
University of North Carolina
Ligand
BDBM82269
((+)-alpha-Propoxyphene | CAS_469-62-5 | PROPOXYPHE...)
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Affinity Data
EC50: 1.50E+4nM
pH: 7.4 T: 2°C
Assay Description:
HTLA cells (HEK-T cells stably expressing a β-arrestin2-TEV fusion protein and a tTa-dependent luciferase reporter) were maintained in DMEM (Cor...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
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ChEBI
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In Depth
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Target
Mas-related G-protein coupled receptor member X2
(Homo sapiens (Human))
University of North Carolina
Ligand
BDBM82269
((+)-alpha-Propoxyphene | CAS_469-62-5 | PROPOXYPHE...)
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Affinity Data
EC50: 3.20E+4nM
pH: 7.4 T: 2°C
Assay Description:
MRGPRX2 stable cells were maintained in DMEM containing 10% FBS, 100 μg/ml hygromycin B, and 15 μg/ml blasticidin. For the calcium mobiliza...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
Purchase
ChEBI
DrugBank
PC cid
PC sid
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In Depth
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Article
PubMed
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