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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 13 hits in this display   

TargetCarbonic anhydrase(Candida albicans (Yeast))
Università

Curated by ChEMBL
LigandPNGBDBM50257201(CHEMBL500826 | sodium propionate)
Affinity DataKi:  5.15E+4nMAssay Description:Inhibition of Candida albicans Nce103More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase [110-330](Flaveria bidentis (Coastal plain yellowtops))
Istituto Di Biostrutture E Bioimmagini-Cnr

LigandPNGBDBM50257201(CHEMBL500826 | sodium propionate)
Affinity DataKi:  9.10E+4nM ΔG°:  -22.7kJ/molepH: 8.3 T: 2°CAssay Description:Inhibition constants of carboxylate inhibitors against F. bidentis CA I were determined by a stopped flow CO2 hydration assay at 20 °C.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 20(Mus musculus)
University Of California

Curated by ChEMBL
LigandPNGBDBM50082199(CH3-CH2-COOH | CHEMBL14021 | Propionsaeure | acide...)
Affinity DataKi:  2.82E+5nMAssay Description:Inhibition of mouse Oat6-mediated [3H]ES uptake in Xenopus oocytes after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50257201(CHEMBL500826 | sodium propionate)
Affinity DataKi:  9.60E+5nMAssay Description:Inhibition of human carbonic anhydrase2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50257201(CHEMBL500826 | sodium propionate)
Affinity DataKi:  1.01E+6nMAssay Description:Inhibition of human cytosolic carbonic anhydrase 1 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 6(Mus musculus)
University Of California

Curated by ChEMBL
LigandPNGBDBM50082199(CH3-CH2-COOH | CHEMBL14021 | Propionsaeure | acide...)
Affinity DataKi:  8.18E+6nMAssay Description:Inhibition of mouse Oat1-mediated [3H]PAH uptake in Xenopus oocytes after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50082199(CH3-CH2-COOH | CHEMBL14021 | Propionsaeure | acide...)
Affinity DataIC50:  1.30E+5nMAssay Description:Agonist activity at human FFA2 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 3(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50082199(CH3-CH2-COOH | CHEMBL14021 | Propionsaeure | acide...)
Affinity DataEC50:  1.17E+4nMAssay Description:Agonist activity at human FFA3 receptor stably expressed in Flp-In T-Rex HEK293 cells cotransfected with eYFP assessed as inhibition of forskolin-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50082199(CH3-CH2-COOH | CHEMBL14021 | Propionsaeure | acide...)
Affinity DataEC50:  2.57E+5nMAssay Description:Agonist activity at human FFA2R expressed in CHOK1 cells assessed as induction of GTPgamma35S binding preincubated for 15 mins followed by GTPgamma35...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 2(Mus musculus)
University Of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50082199(CH3-CH2-COOH | CHEMBL14021 | Propionsaeure | acide...)
Affinity DataEC50:  2.51E+5nMAssay Description:Agonist activity at FFA2R in mouse mature adipocytes assessed as inhibition of isoproterenol-induced glycerol productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 3(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50082199(CH3-CH2-COOH | CHEMBL14021 | Propionsaeure | acide...)
Affinity DataEC50:  1.20E+4nMAssay Description:Agonist activity at human GPCR41 transfected in HEK293 cells assessed as [35S]GTPgammaS binding by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 3(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50082199(CH3-CH2-COOH | CHEMBL14021 | Propionsaeure | acide...)
Affinity DataEC50:  1.07E+4nMAssay Description:Agonist activity at human FFA3 receptor stably expressed in Flp-In T-Rex HEK293 cell membrane assessed as stimulation of [35S]-GTPgammaS binding meas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50082199(CH3-CH2-COOH | CHEMBL14021 | Propionsaeure | acide...)
Affinity DataEC50:  2.50E+5nMAssay Description:Agonist activity at human GPCR43 transfected in HEK293 cells assessed as [35S]GTPgammaS binding by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed