Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 4 hits in this display
BDBM301453(7-{1-[1-(2,5-difluorophenyl)-1H-1,2,3-triazol-4-yl...)
BDBM301453(7-{1-[1-(2,5-difluorophenyl)-1H-1,2,3-triazol-4-yl...)
BDBM301453(7-{1-[1-(2,5-difluorophenyl)-1H-1,2,3-triazol-4-yl...)
EC50: 9.95nMAssay Description:Primary cystic fibrosis human bronchial epithelial (CF hBE) cells were expanded and cultured according to published methods (Neuberger et al., Ch. 4 ...More data for this Ligand-Target Pair
BDBM301453(7-{1-[1-(2,5-difluorophenyl)-1H-1,2,3-triazol-4-yl...)
EC50: 253nMAssay Description:Fischer rat thyroid (FRT) cell lines stably expressing recombinant F508del V470 CFTR and halide-sensitive yellow fluorescent protein (Pedemonte et al...More data for this Ligand-Target Pair