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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetCathepsin G(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50266989(CHEMBL4081142)
Affinity DataKi:  1.70nMAssay Description:Inhibition of human cathepsin G using Suc-AAPF-MCA as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Rattus norvegicus)
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50266989(CHEMBL4081142)
Affinity DataKi:  7.70nMAssay Description:Inhibition of rat mast cell chymase using Suc-AAPF-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50266989(CHEMBL4081142)
Affinity DataKi:  130nMAssay Description:Inhibition of recombinant KLK7 (unknown origin) expressed in zymogen form in Pichia pastorisstrain X-33 using KHLY-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50266989(CHEMBL4081142)
Affinity DataKi:  8.90E+3nMAssay Description:Inhibition of human neutrophil elastase using Suc(OMe)-AAPV-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50266989(CHEMBL4081142)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human PR3 using Suc(OMe)-AAPV-MCA as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed