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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 11 hits in this display   

TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Hokuriku University

LigandPNGBDBM18363((2R,3R,4R,5S,6R)-2-(hydroxymethyl)-6-octylpiperidi...)
Affinity DataKi:  280nM ΔG°:  -38.9kJ/mole IC50:  500nMpH: 5.5 T: 2°CAssay Description:Enzyme activity was determined as the production of fluorescent 4-MU from the substrate. The fluorescence was measured (excitation 362 nm, emission 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50156356(2-Hydroxymethyl-6-octyl-piperidine-3,4,5-triol | C...)
Affinity DataIC50:  90nMAssay Description:Inhibition of rat intestinal isomaltase using disaccharideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM18363((2R,3R,4R,5S,6R)-2-(hydroxymethyl)-6-octylpiperidi...)
Affinity DataIC50:  120nMAssay Description:Inhibition of rat intestinal isomaltase using isomoltose as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative alpha-glucosidase(Oryza sativa subsp. japonica)
Universit£

Curated by ChEMBL
LigandPNGBDBM50156356(2-Hydroxymethyl-6-octyl-piperidine-3,4,5-triol | C...)
Affinity DataIC50:  590nMAssay Description:Inhibitory activity against alpha-Glucosidase from riceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50156356(2-Hydroxymethyl-6-octyl-piperidine-3,4,5-triol | C...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of rat intestinal sucrase using disaccharideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM18363((2R,3R,4R,5S,6R)-2-(hydroxymethyl)-6-octylpiperidi...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of rat intestinal sucrase using sucrose as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50156356(2-Hydroxymethyl-6-octyl-piperidine-3,4,5-triol | C...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of rat intestinal maltase using disaccharideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal alpha-glucosidase(Rattus norvegicus)
University Of Toyama

Curated by ChEMBL
LigandPNGBDBM18363((2R,3R,4R,5S,6R)-2-(hydroxymethyl)-6-octylpiperidi...)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of rat intestinal maltase using moltose as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-lysine 6-oxidase(Homo sapiens (Human))
Hokuriku University

LigandPNGBDBM18363((2R,3R,4R,5S,6R)-2-(hydroxymethyl)-6-octylpiperidi...)
Affinity DataIC50:  5.00E+3nMpH: 4.5 T: 2°CAssay Description:Enzyme activity was determined as the production of fluorescent 4-MU from the substrate. The fluorescence was measured (excitation 362 nm, emission 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-glucosidase(Prunus avium)
Universit£

Curated by ChEMBL
LigandPNGBDBM50156356(2-Hydroxymethyl-6-octyl-piperidine-3,4,5-triol | C...)
Affinity DataIC50:  2.70E+4nMAssay Description:Inhibitory activity against beta-Glucosidase from sweet almondMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-glucosidase A(Caldocellum saccharolyticum)
Universit£

Curated by ChEMBL
LigandPNGBDBM50156356(2-Hydroxymethyl-6-octyl-piperidine-3,4,5-triol | C...)
Affinity DataIC50:  1.10E+5nMAssay Description:Inhibitory activity against beta-Glucosidase from Caldocellum saccharolyticumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed