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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetCytochrome P450 3A2(RAT)
Qingdao University Medical College

Curated by ChEMBL
LigandPNGBDBM50592756(CHEMBL5182450)
Affinity DataKi:  5.26E+4nMAssay Description:Inhibition of CYP3A2 in rat liver microsomes using midazolam as substrateMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCytochrome P450 1A2(Rattus norvegicus)
Qingdao University Medical College

Curated by ChEMBL
LigandPNGBDBM50592756(CHEMBL5182450)
Affinity DataKi:  1.27E+5nMAssay Description:Inhibition of CYP1A2 in rat liver microsomes using phenacetin as substrateMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCytochrome P450 2D1(Rattus norvegicus)
Qingdao University Medical College

Curated by ChEMBL
LigandPNGBDBM50592756(CHEMBL5182450)
Affinity DataKi:  1.79E+5nMAssay Description:Inhibition of CYP2D1 in rat liver microsomes using dextromethorphan as substrateMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCytochrome P450 2E1(Rattus norvegicus (rat))
Qingdao University Medical College

Curated by ChEMBL
LigandPNGBDBM50592756(CHEMBL5182450)
Affinity DataKi:  1.96E+5nMAssay Description:Inhibition of CYP2E1 in rat liver microsomes using chlorzoxazone as substrateMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCytochrome P450 2C6(Rattus norvegicus)
Qingdao University Medical College

Curated by ChEMBL
LigandPNGBDBM50592756(CHEMBL5182450)
Affinity DataKi:  2.03E+5nMAssay Description:Inhibition of CYP2C6 in rat liver microsomes using diclofenac as substrateMore data for this Ligand-Target Pair
In DepthDetails PubMed