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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50101598(CHEMBL307495 | [3-Carboxy-2-(dodecane-1-sulfonylam...)
Affinity DataIC50:  700nMAssay Description:Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]-palmitoyl-CoA radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50101598(CHEMBL307495 | [3-Carboxy-2-(dodecane-1-sulfonylam...)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibitory activity against rat heart mitochondrial carnitine palmitoyltransferase 1b using [14C]-palmitoyl-CoA as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50101598(CHEMBL307495 | [3-Carboxy-2-(dodecane-1-sulfonylam...)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I from rat liver mitochondriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50101598(CHEMBL307495 | [3-Carboxy-2-(dodecane-1-sulfonylam...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed