Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetCysteinyl leukotriene receptor 1/2(Homo sapiens (Human))
TBA

Curated by ChEMBL

LigandBDBM50021025(3-[(2-Carboxy-ethylsulfanyl)-(2-dodecyl-phenyl)-me...)Copy SMILESCopy InChI

Affinity DataKi:  445nMAssay Description:Compound is evaluated for its ability to inhibit [3H]LTD4 binding to Cysteinyl leukotriene D4 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
antibodypediaantibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidPatentsSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
TBA

Curated by ChEMBL

LigandBDBM50021025(3-[(2-Carboxy-ethylsulfanyl)-(2-dodecyl-phenyl)-me...)Copy SMILESCopy InChI

Affinity DataKi:  445nMAssay Description:Binding constant was determined as affinity to displace [3H]-LTD4 from Cysteinyl leukotriene D4 receptor on guinea pig lung membraneMore data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidPatentsSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI