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Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
9
hits in this display
Target
Lysine-specific demethylase 4C
(Homo sapiens (Human))
University Of Oxford
Curated by
ChEMBL
Ligand
BDBM50158888
(CHEMBL3785984)
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Affinity Data
IC50: 3.90E+3nM
Assay Description:
Inhibition of KDM4C (unknown origin) using H3K9me3 as substrate after 24 hrs by alphascreen assay
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Target
Lysine-specific demethylase 4E
(Homo sapiens (Human))
University Of Oxford
Curated by
ChEMBL
Ligand
BDBM50158888
(CHEMBL3785984)
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Affinity Data
IC50: 4.50E+4nM
Assay Description:
Inhibition of KDM4E (unknown origin) after 24 hrs by alphascreen assay
More data for this Ligand-Target Pair
Target Info
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MMDB
KEGG
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Target
Lysine-specific demethylase 3A
(Homo sapiens (Human))
University Of Oxford
Curated by
ChEMBL
Ligand
BDBM50158888
(CHEMBL3785984)
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Affinity Data
IC50: >1.00E+5nM
Assay Description:
Inhibition of KDM3A (unknown origin) after 24 hrs by alphascreen assay
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Target
Lysine-specific demethylase 2A
(Homo sapiens (Human))
University Of Oxford
Curated by
ChEMBL
Ligand
BDBM50158888
(CHEMBL3785984)
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Affinity Data
IC50: >1.00E+5nM
Assay Description:
Inhibition of KDM2A (unknown origin) after 24 hrs by alphascreen assay
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Target
Prolyl 4-hydroxylase
(Paramecium bursaria Chlorella virus 1)
University Of Oxford
Curated by
ChEMBL
Ligand
BDBM50158888
(CHEMBL3785984)
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Affinity Data
IC50: >1.00E+5nM
Assay Description:
Inhibition of N-terminal His6-tagged recombinant Paramecium bursaria chlorella virus 1 CPH expressed in Escherichia coli Rosetta 2 (DE3) cells pre-in...
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Target Info
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Target
Lysine-specific demethylase 5C
(Homo sapiens (Human))
University Of Oxford
Curated by
ChEMBL
Ligand
BDBM50158888
(CHEMBL3785984)
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Affinity Data
IC50: >1.00E+5nM
Assay Description:
Inhibition of KDM5C (unknown origin) after 24 hrs by alphascreen assay
More data for this Ligand-Target Pair
Target Info
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MMDB
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KEGG
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Target
Lysine-specific demethylase 6B
(Homo sapiens (Human))
University Of Oxford
Curated by
ChEMBL
Ligand
BDBM50158888
(CHEMBL3785984)
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Affinity Data
IC50: >1.00E+5nM
Assay Description:
Inhibition of KDM6B (unknown origin) after 24 hrs by alphascreen assay
More data for this Ligand-Target Pair
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Target
Egl nine homolog 1
(Homo sapiens (Human))
University Of Oxford
Curated by
ChEMBL
Ligand
BDBM50158888
(CHEMBL3785984)
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Affinity Data
IC50: >1.00E+5nM
Assay Description:
Inhibition of PHD2 catalytic domain (unknown origin) after 24 hrs by alphascreen assay
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
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KEGG
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Target
Lysine-specific demethylase 4A
(Homo sapiens (Human))
University Of Oxford
Curated by
ChEMBL
Ligand
BDBM50158888
(CHEMBL3785984)
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Affinity Data
EC50: 3.80E+3nM
Assay Description:
Inhibition of human Flag-tagged KDM4A expressed in human HeLa cells assessed as increase in H3K9me3 level after 24 hrs by DAPI staining based immunof...
More data for this Ligand-Target Pair
Target Info
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antibodypedia
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CHEMBL
PC cid
PC sid
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PubMed
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