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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 9 hits in this display   

TargetLysine-specific demethylase 4C(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50158888(CHEMBL3785984)
Affinity DataIC50:  3.90E+3nMAssay Description:Inhibition of KDM4C (unknown origin) using H3K9me3 as substrate after 24 hrs by alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 4E(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50158888(CHEMBL3785984)
Affinity DataIC50:  4.50E+4nMAssay Description:Inhibition of KDM4E (unknown origin) after 24 hrs by alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 3A(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50158888(CHEMBL3785984)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of KDM3A (unknown origin) after 24 hrs by alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 2A(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50158888(CHEMBL3785984)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of KDM2A (unknown origin) after 24 hrs by alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl 4-hydroxylase(Paramecium bursaria Chlorella virus 1)
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50158888(CHEMBL3785984)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of N-terminal His6-tagged recombinant Paramecium bursaria chlorella virus 1 CPH expressed in Escherichia coli Rosetta 2 (DE3) cells pre-in...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 5C(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50158888(CHEMBL3785984)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of KDM5C (unknown origin) after 24 hrs by alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 6B(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50158888(CHEMBL3785984)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of KDM6B (unknown origin) after 24 hrs by alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEgl nine homolog 1(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50158888(CHEMBL3785984)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of PHD2 catalytic domain (unknown origin) after 24 hrs by alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 4A(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50158888(CHEMBL3785984)
Affinity DataEC50:  3.80E+3nMAssay Description:Inhibition of human Flag-tagged KDM4A expressed in human HeLa cells assessed as increase in H3K9me3 level after 24 hrs by DAPI staining based immunof...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed