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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
7
hits in this display
Target
Lysine-specific demethylase 5B
(Homo sapiens (Human))
Kyoto Prefectural University Of Medicine
Curated by
ChEMBL
Ligand
BDBM50532176
(CHEMBL4542928)
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Affinity Data
IC50: 1.30nM
Assay Description:
Inhibition of human N-terminal FLAG/His-tagged KDM5B (2 to 751 residues) expressed in baculovirus infected Sf9 insect cells using H3(1-21)K4(Me3)-GGK...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
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Article
PubMed
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Target
Lysine-specific demethylase 5A
(Homo sapiens (Human))
Kyoto Prefectural University Of Medicine
Curated by
ChEMBL
Ligand
BDBM50532176
(CHEMBL4542928)
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Copy InChI
Affinity Data
IC50: 4.40nM
Assay Description:
Inhibition of human C-terminal FLAG-tagged KDM5A (1 to 1090 residues) expressed in baculovirus infected Sf9 insect cells using H3(1-21)K4(Me3)-GGK(Bi...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
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Target
Lysine-specific demethylase 5C
(Homo sapiens (Human))
Kyoto Prefectural University Of Medicine
Curated by
ChEMBL
Ligand
BDBM50532176
(CHEMBL4542928)
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Affinity Data
IC50: 6.20nM
Assay Description:
Inhibition of full-length human N-terminal FLAG/His-tagged KDM5C (2 to 1560 residues) expressed in baculovirus infected Sf9 insect cells using H3(1-2...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
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Target
Lysine-specific demethylase 3A
(Homo sapiens (Human))
Kyoto Prefectural University Of Medicine
Curated by
ChEMBL
Ligand
BDBM50532176
(CHEMBL4542928)
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Affinity Data
IC50: 5.00E+4nM
Assay Description:
Inhibition of human N-terminal FLAG-tagged KDM3A (2 to 1321 residues) expressed in baculovirus infected Sf9 insect cells using H3(1-21)K9(Me1)-GGK(Bi...
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
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Target
Lysine-specific demethylase 6B
(Homo sapiens (Human))
Kyoto Prefectural University Of Medicine
Curated by
ChEMBL
Ligand
BDBM50532176
(CHEMBL4542928)
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Affinity Data
IC50: >5.00E+4nM
Assay Description:
Inhibition of human C-terminal FLAG-tagged KDM6B (1043 to end residues) expressed in baculovirus infected Sf9 insect cells using H3(21-44)-K27(Me3)-G...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
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Target
Lysine-specific demethylase 2A
(Homo sapiens (Human))
Kyoto Prefectural University Of Medicine
Curated by
ChEMBL
Ligand
BDBM50532176
(CHEMBL4542928)
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Affinity Data
IC50: >5.00E+4nM
Assay Description:
Inhibition of human N-terminal FLAG/Avi-tagged KDM2A (2 to 700 residues) expressed in baculovirus infected Sf9 insect cells using H3(21-44)-K36(Me2)-...
More data for this Ligand-Target Pair
Target Info
PDB
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UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
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PC sid
In Depth
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Article
PubMed
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Target
Histone lysine demethylase PHF8
(Homo sapiens (Human))
Kyoto Prefectural University Of Medicine
Curated by
ChEMBL
Ligand
BDBM50532176
(CHEMBL4542928)
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Affinity Data
IC50: >5.00E+4nM
Assay Description:
Inhibition of human N-terminal FLAG-tagged KDM7B (2 to 525 residues) expressed in baculovirus infected Sf9 insect cells using H3(1-21)K9(Me2)-GGK(Bio...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI