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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 7 hits in this display   

Target72 kDa type IV collagenase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50294123(2-(4'-Butoxy-N-isopropoxybiphenyl-4-ylsulfonamido)...)
Affinity DataIC50:  5.5nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50294123(2-(4'-Butoxy-N-isopropoxybiphenyl-4-ylsulfonamido)...)
Affinity DataIC50:  15nMAssay Description:Inhibition of MMP13-mediated collagen degradation by SDS-PAGEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50294123(2-(4'-Butoxy-N-isopropoxybiphenyl-4-ylsulfonamido)...)
Affinity DataIC50:  44nMAssay Description:Inhibition of MMP9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil collagenase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50294123(2-(4'-Butoxy-N-isopropoxybiphenyl-4-ylsulfonamido)...)
Affinity DataIC50:  560nMAssay Description:Inhibition of MMP8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50294123(2-(4'-Butoxy-N-isopropoxybiphenyl-4-ylsulfonamido)...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of MMP3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-14(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50294123(2-(4'-Butoxy-N-isopropoxybiphenyl-4-ylsulfonamido)...)
Affinity DataIC50:  5.50E+3nMAssay Description:Inhibition of human recombinant MMP14More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50294123(2-(4'-Butoxy-N-isopropoxybiphenyl-4-ylsulfonamido)...)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of MMP1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed