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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 9 hits in this display   

TargetNeutrophil collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50102483(2-(1-((2-methoxyethoxy)carbonyl)piperidin-4-yl)-2-...)
Affinity DataIC50:  294nMAssay Description:Inhibitory activity against matrix metalloprotease-8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50102483(2-(1-((2-methoxyethoxy)carbonyl)piperidin-4-yl)-2-...)
Affinity DataIC50:  295nMAssay Description:Inhibition of MMP8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50102483(2-(1-((2-methoxyethoxy)carbonyl)piperidin-4-yl)-2-...)
Affinity DataIC50:  549nMAssay Description:In vitro inhibitory activity against matrix metalloprotease-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50102483(2-(1-((2-methoxyethoxy)carbonyl)piperidin-4-yl)-2-...)
Affinity DataIC50:  678nMAssay Description:In vitro inhibitory activity against matrix metalloprotease-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50102483(2-(1-((2-methoxyethoxy)carbonyl)piperidin-4-yl)-2-...)
Affinity DataIC50:  791nMAssay Description:In vitro inhibitory activity against matrix metalloprotease-13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50102483(2-(1-((2-methoxyethoxy)carbonyl)piperidin-4-yl)-2-...)
Affinity DataIC50:  794nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50102483(2-(1-((2-methoxyethoxy)carbonyl)piperidin-4-yl)-2-...)
Affinity DataIC50:  2.99E+3nMAssay Description:In vitro inhibition of human matrix metalloprotease-9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrilysin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50102483(2-(1-((2-methoxyethoxy)carbonyl)piperidin-4-yl)-2-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity against matrix metalloprotease-7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50102483(2-(1-((2-methoxyethoxy)carbonyl)piperidin-4-yl)-2-...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibitory activity against matrix metalloprotease-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed