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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetPoly [ADP-ribose] polymerase tankyrase-1(Homo sapiens (Human))
Lauren Mccallister

Curated by ChEMBL
LigandPNGBDBM50544641(CHEMBL4645574)
Affinity DataIC50:  0.260nMAssay Description:Inhibition of human GST-tagged tankyrase 1 autophosphorylation by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
Lauren Mccallister

Curated by ChEMBL
LigandPNGBDBM50544641(CHEMBL4645574)
Affinity DataIC50:  0.440nMAssay Description:Inhibition of human GST-tagged tankyrase 2 autophosphorylationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed