Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 57 hits in this display
BDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
BDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
BDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
BDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
BDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
BDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
BDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
BDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
BDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
BDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
BDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
Carbamate kinase(Giardia intestinalis)Commonwealth Scientific And Industrial Research Organization
Curated by ChEMBL
BDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
BDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
BDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
BDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
BDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
IC50: 1.04E+3nMAssay Description:Inhibition of SARS-CoV-2 3CL protease using Dabcyl-KNSTLQSGLRKE-Edan as substrate incubated for 30 mins and measured by FRET assayMore data for this Ligand-Target Pair
BDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
BDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
BDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
BDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
BDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
BDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
BDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
BDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
BDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
BDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
Caspase-1(Homo sapiens (Human))Depaul University
BDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
BDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
BDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
BDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
IC50: 3.00E+3nMAssay Description:Inhibition of NLRP3 in mouse J774A.1 cells infected with FLA-ST assessed as inhibition of LPS- induced IL-1beta production by ELISAMore data for this Ligand-Target Pair
BDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
BDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
BDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
IC50: 6.72E+3nMAssay Description:Inhibition of SARS-CoV 3CL protease using Dabcyl-KNSTLQSGLRKE-Edan as substrate incubated for 30 mins and measured by FRET assayMore data for this Ligand-Target Pair
BDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
BDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
BDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
BDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
BDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
BDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
BDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
BDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
BDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
BDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
BDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
BDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
BDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
Replicase polyprotein 1ab(Human SARS coronavirus (SARS-CoV) (Severe acute re...)Fraunhofer Institute For Translational Medicine and Pharmacology (Itmp) and Fraunhofer Cluster of Excellence For Immune Mediated Diseases (Cimd
BDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
IC50: 2.68E+4nMAssay Description:Primary assay principle based on quenched FRET peptide substrate of SARS-CoV-2 3CL-Pro (lhs). Inhibiting compounds reduce fluorescence signal relativ...More data for this Ligand-Target Pair
BDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
BDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
BDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
BDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
BDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
BDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
BDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
BDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
BDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
EC50: 3.00E+3nMAssay Description:Agonist activity at human TRPA1 channel expressed in CHO cells assessed as increase in intracellular calcium levelsMore data for this Ligand-Target Pair
BDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
Displayed 1 to 50 (of 57 total ) | Next | Last >>