Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 1 hits in this display   

TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Rccs Istituto Giannina Gaslini

Curated by ChEMBL
LigandPNGBDBM50546507(CHEMBL4746459)
Affinity DataEC50:  3.20E+3nMAssay Description:Potentiation of CFTR F508 deletion mutant (unknown origin) expressed in CFBE41o- cells coexpressing HS-YFP assessed as increase in intracellular cAMP...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed