Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetGamma-aminobutyric acid receptor subunit alpha-5(Homo sapiens (Human))
Moltech

Curated by ChEMBL
LigandPNGBDBM50244262(CHEMBL471978 | ethyl 7-ethynyl-4-methyl-5-oxo-4,5-...)
Affinity DataKi:  1.68nMAssay Description:Binding affinity to GABAA alpha-5-beta-3-gamma-2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-2(Homo sapiens (Human))
Moltech

Curated by ChEMBL
LigandPNGBDBM50244262(CHEMBL471978 | ethyl 7-ethynyl-4-methyl-5-oxo-4,5-...)
Affinity DataKi:  21.4nMAssay Description:Binding affinity to GABAA alpha-2-beta-3-gamma-2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
Moltech

Curated by ChEMBL
LigandPNGBDBM50244262(CHEMBL471978 | ethyl 7-ethynyl-4-methyl-5-oxo-4,5-...)
Affinity DataKi:  28.4nMAssay Description:Binding affinity to GABAA alpha-1-beta-3-gamma-2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-6(Homo sapiens (Human))
Moltech

Curated by ChEMBL
LigandPNGBDBM50244262(CHEMBL471978 | ethyl 7-ethynyl-4-methyl-5-oxo-4,5-...)
Affinity DataKi: >100nMAssay Description:Binding affinity to GABAA alpha-6-beta-3-gamma-2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3(Homo sapiens (Human))
Moltech

Curated by ChEMBL
LigandPNGBDBM50244262(CHEMBL471978 | ethyl 7-ethynyl-4-methyl-5-oxo-4,5-...)
Affinity DataKi:  198nMAssay Description:Binding affinity to GABAA alpha-3-beta-3-gamma-2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed