Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Homo sapiens (Human))
Nippon Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50218691(CHEMBL51667)
Affinity DataIC50:  4.30nMAssay Description:Compound was evaluated for its Beta adrenergic receptor blocking actionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1/2(Homo sapiens (Human))
Nippon Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50218691(CHEMBL51667)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibitory activity against Candida albicans N-myristoyltransferase (CaNmt)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1/2(Homo sapiens (Human))
Nippon Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50218691(CHEMBL51667)
Affinity DataIC50:  4.70E+5nMAssay Description:Inhibitory activity against human N-myristoyltransferase (HsNmt)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycylpeptide N-tetradecanoyltransferase(Candida albicans (Yeast))TBA
LigandPNGBDBM50218691(CHEMBL51667)
Affinity DataIC50:  8.33E+8nMAssay Description:Inhibition of candida N-myristoyltransferaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGlycylpeptide N-tetradecanoyltransferase(Candida albicans (Yeast))TBA
LigandPNGBDBM50218691(CHEMBL51667)
Affinity DataIC50:  8.33E+8nMAssay Description:Inhibition of candida N-myristoyltransferaseMore data for this Ligand-Target Pair
In DepthDetails Article