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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 9 hits in this display   

TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM23771((3-{[1-benzyl-3-(carbamoylmethyl)-2-ethyl-1H-indol...)
Affinity DataIC50:  23nMAssay Description:Inhibition of human non-pancreatic secretory phospholipase A2 (PLA2) in a chromogenic assayMore data for this Ligand-Target Pair
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM23771((3-{[1-benzyl-3-(carbamoylmethyl)-2-ethyl-1H-indol...)
Affinity DataIC50:  470nMAssay Description:Inhibition of human recombinant group 2A phospholipase A2 by fluorimetric assayMore data for this Ligand-Target Pair
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM23771((3-{[1-benzyl-3-(carbamoylmethyl)-2-ethyl-1H-indol...)
Affinity DataIC50:  470nMAssay Description:Inhibition of human group IIA PLA2 by fluorimetric assayMore data for this Ligand-Target Pair
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM23771((3-{[1-benzyl-3-(carbamoylmethyl)-2-ethyl-1H-indol...)
Affinity DataIC50:  470nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
TargetPhospholipase A2, major isoenzyme(Sus scrofa (pig))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23771((3-{[1-benzyl-3-(carbamoylmethyl)-2-ethyl-1H-indol...)
Affinity DataIC50:  8.00E+3nMAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue as the substrate. The increase in fluorescence (ex @342 nm and em@388 nm) of the enzy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, major isoenzyme(Sus scrofa (pig))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23771((3-{[1-benzyl-3-(carbamoylmethyl)-2-ethyl-1H-indol...)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of pig group IB PLA2 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, major isoenzyme(Sus scrofa (pig))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23771((3-{[1-benzyl-3-(carbamoylmethyl)-2-ethyl-1H-indol...)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of porcine group 1B phospholipase A2 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM23771((3-{[1-benzyl-3-(carbamoylmethyl)-2-ethyl-1H-indol...)
Affinity DataIC50:  3.55E+4nMAssay Description:Inhibitory activity against porcine pancreatic Phospholipase A2More data for this Ligand-Target Pair
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM23771((3-{[1-benzyl-3-(carbamoylmethyl)-2-ethyl-1H-indol...)
Affinity DataIC50:  9.11E+4nMAssay Description:Inhibitory activity against human pancreatic Phospholipase A2More data for this Ligand-Target Pair