Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 15 hits in this display
IC50: >2.50E+4nMAssay Description:Inhibition of Aurora B kinase in human HeLa Kyoto cells assessed as effect on distribution of phspho-histone H3 ser10 level incubated for 20 hrsMore data for this Ligand-Target Pair
Kd: 450nMAssay Description:Binding affinity to human DAPK2 expressed in Escherichia coli BL21 cells incubated for 1 hr by active site directed binding competition assayMore data for this Ligand-Target Pair
Kd: 480nMAssay Description:Binding affinity to human PIP5K2C expressed in Escherichia coli BL21 cells incubated for 1 hr by active site directed binding competition assayMore data for this Ligand-Target Pair
Kd: 2.90E+3nMAssay Description:Binding affinity to human YSK4 expressed in Escherichia coli BL21 cells incubated for 1 hr by active site directed binding competition assayMore data for this Ligand-Target Pair
Kd: 1.50E+3nMAssay Description:Binding affinity to human PIK3CG expressed in Escherichia coli BL21 cells incubated for 1 hr by active site directed binding competition assayMore data for this Ligand-Target Pair
EC50: 6.00E+3nMAssay Description:Inhibition of Aurora A kinase in human HeLa Kyoto cells assessed as induction of defective chromosome alignment during metaphase incubated for 20 hrsMore data for this Ligand-Target Pair