Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 6 hits in this display
BDBM278129(5-(4-((1-ethyl-1H-pyrazol-4-yl)amino)-1,3,5-triazi...)
BDBM278129(5-(4-((1-ethyl-1H-pyrazol-4-yl)amino)-1,3,5-triazi...)
IC50: 9nMAssay Description:Enzymatic activity of IKKε and TBK1 was measured using a homogeneous time resolved fluorescence resonance energy transfer (TR-FRET) assay that m...More data for this Ligand-Target Pair
BDBM278129(5-(4-((1-ethyl-1H-pyrazol-4-yl)amino)-1,3,5-triazi...)
BDBM278129(5-(4-((1-ethyl-1H-pyrazol-4-yl)amino)-1,3,5-triazi...)
BDBM278129(5-(4-((1-ethyl-1H-pyrazol-4-yl)amino)-1,3,5-triazi...)
IC50: 9.00E+3nMpH: 7.0Assay Description:Enzymatic activity of IKKε and TBK1 was measured using a homogeneous time resolved fluorescence resonance energy transfer (TR-FRET) assay that m...More data for this Ligand-Target Pair
BDBM278129(5-(4-((1-ethyl-1H-pyrazol-4-yl)amino)-1,3,5-triazi...)