Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 8 hits in this display
BDBM454346(US10717734, Compound 22 | US10717734, Compound 23)
BDBM454346(US10717734, Compound 22 | US10717734, Compound 23)
BDBM454346(US10717734, Compound 22 | US10717734, Compound 23)
IC50: >3.00E+3nMAssay Description:SSAO/VAP-1: Human recombinant SSAO/VAP-1 amine oxidase activity was determined using the coupled colorimetric method as described for monoamine oxida...More data for this Ligand-Target Pair
BDBM454346(US10717734, Compound 22 | US10717734, Compound 23)
IC50: >3.00E+3nMAssay Description:MAO-B: The specificity of the compounds of this invention was tested by determining their ability to inhibit MAO-B activities in vitro. Recombinant h...More data for this Ligand-Target Pair
BDBM454346(US10717734, Compound 22 | US10717734, Compound 23)
BDBM454346(US10717734, Compound 22 | US10717734, Compound 23)
IC50: <3.00E+5nMAssay Description:LOX and LOXL2: Lysyl oxidase (LOX) is an extracellular copper dependent enzyme which oxidizes peptidyl lysine and hydroxylysine residues in collagen ...More data for this Ligand-Target Pair
BDBM454346(US10717734, Compound 22 | US10717734, Compound 23)
IC50: >3.00E+5nMAssay Description:LOX and LOXL2: Lysyl oxidase (LOX) is an extracellular copper dependent enzyme which oxidizes peptidyl lysine and hydroxylysine residues in collagen ...More data for this Ligand-Target Pair
BDBM454346(US10717734, Compound 22 | US10717734, Compound 23)
IC50: <3.00E+5nMAssay Description:LOX and LOXL2: Lysyl oxidase (LOX) is an extracellular copper dependent enzyme which oxidizes peptidyl lysine and hydroxylysine residues in collagen ...More data for this Ligand-Target Pair