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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetAdenosine kinase(Rat)
Abbott Laboratories

LigandPNGBDBM14491(5-(2H-1,3-benzodioxol-5-yl)-6-{2-[4-(dimethylamino...)
Affinity DataIC50:  9nMpH: 7.5 T: 23°CAssay Description:ADK activity was monitored by a radiochemical assay, which measures the conversion of radioactive Ado ([U-14C] adenosine or [2-3H] adenosine) to AMP ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM14491(5-(2H-1,3-benzodioxol-5-yl)-6-{2-[4-(dimethylamino...)
Affinity DataIC50:  9nMAssay Description:Inhibition of cytosolic adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM14491(5-(2H-1,3-benzodioxol-5-yl)-6-{2-[4-(dimethylamino...)
Affinity DataIC50:  250nMAssay Description:Inhibition of adenosine kinase in intact cells assessed as adenosine phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed