Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetA disintegrin and metalloproteinase with thrombospondin motifs 5(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50256700(2-(N-methyl-N-phenylamino)-N-((5-chloro-8-hydroxyq...)
Affinity DataIC50:  560nMAssay Description:Inhibition of ADAMTS5 by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetA disintegrin and metalloproteinase with thrombospondin motifs 4(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50256700(2-(N-methyl-N-phenylamino)-N-((5-chloro-8-hydroxyq...)
Affinity DataIC50: >2.20E+4nMAssay Description:Inhibition of ADAMTS4 by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMacrophage metalloelastase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50256700(2-(N-methyl-N-phenylamino)-N-((5-chloro-8-hydroxyq...)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of MMP12 by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50256700(2-(N-methyl-N-phenylamino)-N-((5-chloro-8-hydroxyq...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of MMP13 by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed