Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 8 hits in this display   

TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
University Of California Riverside

Curated by ChEMBL
LigandPNGBDBM50588301(CHEMBL5195146)
Affinity DataIC50:  266nMAssay Description:Antagonist activity at N-terminal His-tagged cIAP1-BIR3 domain (unknown origin) expressed in Escherichia coli BL21 using AVPIAQKSEK-biotinylated pept...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBaculoviral IAP repeat-containing protein 7(Homo sapiens (Human))
University Of California Riverside

Curated by ChEMBL
LigandPNGBDBM50588301(CHEMBL5195146)
Affinity DataIC50:  278nMAssay Description:Antagonist activity at N-terminal His-tagged wild type ML-IAP BIR domain (63 to 179 residues) (unknown origin) expressed in Escherichia coli BL21 usi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBaculoviral IAP repeat-containing protein 7(Homo sapiens (Human))
University Of California Riverside

Curated by ChEMBL
LigandPNGBDBM50588301(CHEMBL5195146)
Affinity DataIC50:  291nMAssay Description:Antagonist activity at N-terminal His-tagged wild type ML-IAP BIR domain (63 to 179 residues)(unknown origin) expressed in Escherichia coli BL21 usin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetE3 ubiquitin-protein ligase XIAP(Homo sapiens (Human))
University Of California Riverside

Curated by ChEMBL
LigandPNGBDBM50588301(CHEMBL5195146)
Affinity DataIC50:  323nMAssay Description:Antagonist activity at N-terminal His-tagged XIAP-BIR3 domain (253 to 347 residues)(unknown origin) expressed in Escherichia coli BL21 using AVPIAQKS...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
University Of California Riverside

Curated by ChEMBL
LigandPNGBDBM50588301(CHEMBL5195146)
Affinity DataIC50:  370nMAssay Description:Antagonist activity at N-terminal His-tagged cIAP1-BIR3 domain (unknown origin) expressed in Escherichia coli BL21 using AVPIAQKSEK-biotinylated pept...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBaculoviral IAP repeat-containing protein 3(Homo sapiens (Human))
University Of California Riverside

Curated by ChEMBL
LigandPNGBDBM50588301(CHEMBL5195146)
Affinity DataIC50:  397nMAssay Description:Antagonist activity at N-terminal His-tagged cIAP2-BIR3 domain (unknown origin) expressed in Escherichia coli BL21 using AVPIAQKSEK-biotinylated pept...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBaculoviral IAP repeat-containing protein 3(Homo sapiens (Human))
University Of California Riverside

Curated by ChEMBL
LigandPNGBDBM50588301(CHEMBL5195146)
Affinity DataIC50:  530nMAssay Description:Antagonist activity at N-terminal His-tagged cIAP2-BIR3 domain (unknown origin) expressed in Escherichia coli BL21 using AVPIAQKSEK-biotinylated pept...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetE3 ubiquitin-protein ligase XIAP(Homo sapiens (Human))
University Of California Riverside

Curated by ChEMBL
LigandPNGBDBM50588301(CHEMBL5195146)
Affinity DataIC50:  551nMAssay Description:Antagonist activity at N-terminal His-tagged XIAP-BIR3 domain (253 to 347 residues)(unknown origin) expressed in Escherichia coli BL21 using AVPIAQKS...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed