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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 13 hits in this display   

TargetNorepinephrine transporter(RAT)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM82219(CAS_52760-47-1 | CHEMBL38120 | CP-24441 | Tametral...)
Affinity DataKi:  18nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM82219(CAS_52760-47-1 | CHEMBL38120 | CP-24441 | Tametral...)
Affinity DataKi:  150nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM82219(CAS_52760-47-1 | CHEMBL38120 | CP-24441 | Tametral...)
Affinity DataKi:  840nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM82219(CAS_52760-47-1 | CHEMBL38120 | CP-24441 | Tametral...)
Affinity DataKi:  4.70E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTransporter(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM82219(CAS_52760-47-1 | CHEMBL38120 | CP-24441 | Tametral...)
Affinity DataIC50:  18nMAssay Description:Inhibition of norepinephrine uptake in synaptosomal preparation fro rat hypothalamus, using [3H]norepinephrineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM82219(CAS_52760-47-1 | CHEMBL38120 | CP-24441 | Tametral...)
Affinity DataIC50:  40nMAssay Description:Inhibition of norepinephrine uptake in synaptosomal preparation fro rat hypothalamus, using [3H]norepinephrineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM82219(CAS_52760-47-1 | CHEMBL38120 | CP-24441 | Tametral...)
Affinity DataIC50:  150nMAssay Description:Inhibition of norepinephrine uptake in synaptosomal preparation fro rat hypothalamus, using [3H]norepinephrineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM82219(CAS_52760-47-1 | CHEMBL38120 | CP-24441 | Tametral...)
Affinity DataIC50:  210nMAssay Description:Inhibition of dopamine uptake in synaptosomal preparation in rat corpus striatum, using [3H]dopamineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM82219(CAS_52760-47-1 | CHEMBL38120 | CP-24441 | Tametral...)
Affinity DataIC50:  370nMAssay Description:Inhibition of norepinephrine uptake in synaptosomal preparation fro rat hypothalamus, using [3H]norepinephrineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM82219(CAS_52760-47-1 | CHEMBL38120 | CP-24441 | Tametral...)
Affinity DataIC50:  840nMAssay Description:Inhibition of dopamine uptake in synaptosomal preparation in rat corpus striatum, using [3H]dopamineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM82219(CAS_52760-47-1 | CHEMBL38120 | CP-24441 | Tametral...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of norepinephrine uptake in synaptosomal preparation fro rat hypothalamus, using [3H]norepinephrineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM82219(CAS_52760-47-1 | CHEMBL38120 | CP-24441 | Tametral...)
Affinity DataIC50:  1.48E+3nMAssay Description:Inhibition of 5-HT uptake in synaptosomal preparation from rat corpus striatum, using [3H]5-HTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM82219(CAS_52760-47-1 | CHEMBL38120 | CP-24441 | Tametral...)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of 5-HT uptake in synaptosomal preparation from rat corpus striatum, using [3H]5-HTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed