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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 8 hits in this display   

TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Virginia Commonwealth University

Curated by PDSP Ki Database
LigandPNGBDBM50127390(CHEMBL51355 | RTI-147 | [3-(4-Chloro-phenyl)-8-met...)
Affinity DataKi:  1.38nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50127390(CHEMBL51355 | RTI-147 | [3-(4-Chloro-phenyl)-8-met...)
Affinity DataKi:  1.13E+3nMAssay Description:Inhibition of [3H]paroxetine binding at serotonin transporter was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50127390(CHEMBL51355 | RTI-147 | [3-(4-Chloro-phenyl)-8-met...)
Affinity DataKi:  2.37E+3nMAssay Description:Affinity for norepinephrine transporter determined by [3H]nisoxetine displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNorepinephrine transporter(RAT)
Virginia Commonwealth University

Curated by PDSP Ki Database
LigandPNGBDBM50127390(CHEMBL51355 | RTI-147 | [3-(4-Chloro-phenyl)-8-met...)
Affinity DataKi:  3.95E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50127390(CHEMBL51355 | RTI-147 | [3-(4-Chloro-phenyl)-8-met...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Virginia Commonwealth University

Curated by PDSP Ki Database
LigandPNGBDBM50127390(CHEMBL51355 | RTI-147 | [3-(4-Chloro-phenyl)-8-met...)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of [3H]WIN-35428 binding at dopamine transporter was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50127390(CHEMBL51355 | RTI-147 | [3-(4-Chloro-phenyl)-8-met...)
Affinity DataIC50:  3.94E+3nMAssay Description:Inhibition of [3H]nisoxetine binding at norepinephrine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50127390(CHEMBL51355 | RTI-147 | [3-(4-Chloro-phenyl)-8-met...)
Affinity DataIC50:  1.24E+4nMAssay Description:Inhibition of [3H]paroxetine binding at serotonin transporter was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed