Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 6 hits in this display
BDBM162376(US9051329, Example 1 | US9051329, Example 4)
IC50: 27nMAssay Description:Inhibition of human DPP4 preincubated for 30 mins followed by Gly-Pro-AMC addition measured for 50 mins by continuous fluorescence assayMore data for this Ligand-Target Pair
BDBM162376(US9051329, Example 1 | US9051329, Example 4)
BDBM162376(US9051329, Example 1 | US9051329, Example 4)
IC50: >1.00E+5nMAssay Description:Inhibition of FAP (unknown origin) preincubated for 20 mins followed by Nle-Pro-AMC addition measured for 40 mins by continuous fluorescence assayMore data for this Ligand-Target Pair
BDBM162376(US9051329, Example 1 | US9051329, Example 4)
IC50: >1.00E+5nMAssay Description:Inhibition of QPP (unknown origin) preincubated for 30 mins followed by Nle-Pro-AMC addition measured for 50 mins by continuous fluorescence assayMore data for this Ligand-Target Pair
BDBM162376(US9051329, Example 1 | US9051329, Example 4)
IC50: >1.00E+5nMAssay Description:Inhibition of DPP9 (unknown origin) preincubated for 20 mins followed by Gly-Pro-AMC addition measured for 50 mins by continuous fluorescence assayMore data for this Ligand-Target Pair
BDBM162376(US9051329, Example 1 | US9051329, Example 4)