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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
6
hits in this display
Target
Bromodomain-containing protein 4
(Homo sapiens (Human))
West China Hospital Of Sichuan University
Curated by
ChEMBL
Ligand
BDBM50603594
(CHEMBL5205457)
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Affinity Data
IC50: 107nM
Assay Description:
Inhibition of His-tagged full length recombinant BRD4 (unknown origin) (21 to 153 residues) using SGRGK(Ac)GGK(Ac)GLGK(Ac)GGAK(Ac)RHRK(Biotin)-OH as ...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
PubMed
Copy BDB DOI
Target
Bromodomain-containing protein 3
(Homo sapiens (Human))
West China Hospital Of Sichuan University
Curated by
ChEMBL
Ligand
BDBM50603594
(CHEMBL5205457)
Copy SMILES
Copy InChI
Affinity Data
IC50: 502nM
Assay Description:
Inhibition of His-tagged recombinant BRD3 (unknown origin) (11 to 166 residues) using SGRGK(Ac)GGK(Ac)GLGK(Ac)GGAK(Ac)RHRK(Biotin)-OH as substrate me...
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
PubMed
Copy BDB DOI
Target
Bromodomain-containing protein 2
(Homo sapiens (Human))
West China Hospital Of Sichuan University
Curated by
ChEMBL
Ligand
BDBM50603594
(CHEMBL5205457)
Copy SMILES
Copy InChI
Affinity Data
IC50: 718nM
Assay Description:
Inhibition of His-tagged recombinant BRD2 (unknown origin) (11 to 162 residues) using SGRGK(Ac)GGK(Ac)GLGK(Ac)GGAK(Ac)RHRK(Biotin)-OH as substrate me...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
PubMed
Copy BDB DOI
Target
Bromodomain-containing protein 1
(Homo sapiens (Human))
West China Hospital Of Sichuan University
Curated by
ChEMBL
Ligand
BDBM50603594
(CHEMBL5205457)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+3nM
Assay Description:
Inhibition of His-tagged recombinant BRD1 (unknown origin) (11 to 190 residues) using SGRGK(Ac)GGK(Ac)GLGK(Ac)GGAK(Ac)RHRK(Biotin)-OH as substrate me...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
PubMed
Copy BDB DOI
Target
Bromodomain testis-specific protein
(Homo sapiens (Human))
West China Hospital Of Sichuan University
Curated by
ChEMBL
Ligand
BDBM50603594
(CHEMBL5205457)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+3nM
Assay Description:
Inhibition of His-tagged recombinant BRDT (unknown origin) (21 to 153 residues) using SGRGK(Ac)GGK(Ac)GLGK(Ac)GGAK(Ac)RHRK(Biotin)-OH as substrate me...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
PubMed
Copy BDB DOI
Target
Bromodomain and PHD finger-containing protein 3
(Homo sapiens (Human))
West China Hospital Of Sichuan University
Curated by
ChEMBL
Ligand
BDBM50603594
(CHEMBL5205457)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+3nM
Assay Description:
Inhibition of His-tagged recombinant BRPF3 (unknown origin) (11 to 188 residues) using SGRGK(Ac)GGK(Ac)GLGK(Ac)GGAK(Ac)RHRK(Biotin)-OH as substrate m...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
PubMed
Copy BDB DOI