Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50599467(CHEMBL4287375)
Affinity DataIC50:  93nMAssay Description:Inhibition of human Dyrk1AMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50599467(CHEMBL4287375)
Affinity DataIC50:  95nMAssay Description:Inhibition of human N-terminal His6-tagged DYRK1A expressed in Escherichia coli BL21 (DE3) using KKISGRLSPIMTEQ as substrate incubated in presence of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Homo sapiens (Human))
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50599467(CHEMBL4287375)
Affinity DataIC50:  1.51E+3nMAssay Description:Inhibition of Dyrk1B (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 2(Homo sapiens (Human))
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50599467(CHEMBL4287375)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of Dyrk2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed