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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 6 hits in this display   

TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50057728(3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-pyran-...)
Affinity DataKi:  1.60E+5nMAssay Description:Inhibition of rabbit glycogen phosphorylase B enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50147917((R)-3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-py...)
Affinity DataKi:  1.60E+5nMAssay Description:Inhibitory binding constant against glycogen phosphorylase BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50473932(CHEMBL133616)
Affinity DataKi:  1.99E+5nMAssay Description:Inhibitory activity against Pig Skeletal Glycogen Phosphorylase bMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, muscle form(Homo sapiens (Human))
University Of Alcala

Curated by ChEMBL
LigandPNGBDBM50057728(3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-pyran-...)
Affinity DataKi:  3.80E+6nMAssay Description:Inhibitory activity against rabbit muscle glycogen phosphorylaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50147900((S)-3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-py...)
Affinity DataKi:  3.67E+7nMAssay Description:Inhibitory binding constant against glycogen phosphorylase BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50473956(CHEMBL335777)
Affinity DataKi:  3.98E+7nMAssay Description:Inhibitory activity against Pig Skeletal Glycogen Phosphorylase bMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed